Template:SubstanceBox/Cocaine

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SubstanceBox/Cocaine
Cocaine.svg
Chemical Nomenclature
Common names Cocaine, Coke, Coca, Crack, Blow, Girl, White, Snow, Nose Candy, Yayo, Perico,Gear, Chari
Substitutive name Benzoylmethylecgonine
Systematic name Methyl (1R,2R,3S,5S)-3- (Benzoyloxy)-8-methyl-8-azabicyclo[3.2.1] octane-2-carboxylate
Class Membership
Psychoactive class Stimulant, SNDRI
Chemical class Tropane alkaloid
Routes of Administration

WARNING: Always start with lower doses due to differences between individual body weight, tolerance, metabolism, and personal sensitivity. See responsible use section.


Smoked
Dosage
Bioavailability 90%[1]
Threshold 2.5 mg
Light 5 - 15 mg
Common 15 - 30 mg
Strong 30 - 45 mg
Heavy 45 mg +
Duration
Total 5 - 15 minutes
Onset 3 - 5 seconds
Come up 1 - 2 minutes
Peak 2 - 10 minutes
Offset 1 - 5 minutes
Oral
Dosage
Bioavailability 33%[2]
Threshold 13 mg
Light 13 - 75 mg
Common 75 - 150 mg
Strong 150 - 225 mg
Heavy 225 mg +
Duration
Total 120 - 240 minutes
Onset 30 - 40 minutes
Come up 40 - 50 minutes
Peak 60 - 180 minutes
Offset 10 - 25 minutes



Insufflated
Dosage
Bioavailability 60[3]-80%[4]
Threshold 5 mg
Light 10 - 30 mg
Common 30 - 60 mg
Strong 60 - 90 mg
Heavy 90 mg +
Duration
Total 10 - 90 minutes
Onset 3 - 10 minutes
Come up 5 - 12 minutes
Peak 7.5 - 16 minutes
Offset 10 - 25 minutes
After effects Psychological craving and compulsive redosing





Intravenous
Dosage
Bioavailability 100%
Threshold 2 mg
Light 2 - 5 mg
Common 5 - 10 mg
Strong 10 - 15 mg
Heavy 15 mg +
Duration
Total 5 - 15 minutes
Onset 3 - 5 seconds
Come up 1 - 2 minutes
Peak 2 - 10 minutes
Offset 1 - 5 minutes

DISCLAIMER: PW's dosage information is gathered from users and resources for educational purposes only. It is not a recommendation and should be verified with other sources for accuracy.

  1. Roque Bravo, R; Faria, AC; Brito-da-Costa, AM; Carmo, H; Mladěnka, P; Dias da Silva, D; Remião, F; On Behalf Of The Oemonom, Researchers (13 April 2022). "Cocaine: An Updated Overview on Chemistry, Detection, Biokinetics, and Pharmacotoxicological Aspects including Abuse Pattern". Toxins. 14 (4). doi:10.3390/toxins14040278. PMC 9032145Freely accessible Check |pmc= value (help). PMID 35448887. 
  2. Fattinger K, Benowitz NL, Jones RT, Verotta D (July 2000). "Nasal mucosal versus gastrointestinal absorption of nasally administered cocaine". European Journal of Clinical Pharmacology. 56 (4): 305–10. doi:10.1007/s002280000147. PMID 10954344.  Unknown parameter |s2cid= ignored (help)
  3. Barnett, G., Hawks, R., Resnick, R. (March 1981). "Cocaine pharmacokinetics in humans". Journal of Ethnopharmacology. 3 (2–3): 353–366. doi:10.1016/0378-8741(81)90063-5. ISSN 0378-8741. 
  4. Jeffcoat, A. R., Perez-Reyes, M., Hill, J. M., Sadler, B. M., Cook, C. E. (April 1989). "Cocaine disposition in humans after intravenous injection, nasal insufflation (snorting), or smoking". Drug Metabolism and Disposition: The Biological Fate of Chemicals. 17 (2): 153–159. ISSN 0090-9556.